SCHEMBL29965714

SCHEMBL29965714

CN1CCN(C(=O)c2ccc3c(c2)[nH]c(=O)c2ccc(Br)n23)CC1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.51
AURKB Q96GD4 1/20 0.49
KDR P35968 2/20 0.47
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
POLB P06746 3/20 0.46
TSHR P16473 2/20 0.46
THRB P10828 1/20 0.46
RECQL P46063 1/20 0.46
HSD17B10 Q99714 1/20 0.46
HPGD P15428 2/20 0.45
PDGFRB P09619 1/20 0.45
FGFR1 P11362 1/20 0.45
CDK5 Q00535 1/20 0.44
CDK5R1 Q15078 1/20 0.44
HRH4 Q9H3N8 2/20 0.43
HRH3 Q9Y5N1 1/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13056843 0.79 PARP1 (0.80) PARP1AURKBKDRMEN1KMT2A
SCHEMBL28895087 0.79 PARP1 (0.46) PARP1AURKBKMT2AKDM4E
SCHEMBL3600490 0.78 POLB (0.49) PARP1AURKBKDRMEN1KMT2A
SCHEMBL3600486 0.75 PDE9A (0.58) PARP1AURKBKDRMEN1KMT2A
SCHEMBL29965925 0.74 ALDH1A1 (0.55) PARP1AURKBKDRMEN1KMT2A
SCHEMBL28895268 0.74 ALDH1A1 (0.55) PARP1AURKBKDRMEN1KMT2A
SCHEMBL7026634 0.72 PARP1 (0.55) PARP1KDRMEN1KMT2APOLB
SCHEMBL13056827 0.70 PARP1 (0.80) PARP1AURKBMEN1KMT2APOLB
SCHEMBL3595688 0.69 KDR (0.49) PARP1KDRMEN1KMT2APOLB
SCHEMBL29965987 0.69 PDE5A (0.45) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115368362-A Quinoxalinone derivatives as BTK inhibitors and application thereof 华东理工大学 2022-11-22 CN disclosed