SCHEMBL29965987

SCHEMBL29965987

CC(C)(O)c1ccc2c(c1)[nH]c(=O)c1ccc(Br)n12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 4/20 0.45
PDE9A O76083 4/20 0.45
TNKS O95271 14/20 0.43
TNKS2 Q9H2K2 14/20 0.43
PARP1 P09874 13/20 0.43
ADORA3 P0DMS8 1/20 0.43
SLC6A3 Q01959 1/20 0.43
PARP6 Q2NL67 1/20 0.43
PARP10 Q53GL7 1/20 0.43
TIPARP Q7Z3E1 1/20 0.43
PARP8 Q8N3A8 1/20 0.43
PARP12 Q9H0J9 1/20 0.43
PARP11 Q9NR21 1/20 0.43
PARP2 Q9UGN5 1/20 0.43
PARP3 Q9Y6F1 1/20 0.43
TP53 P04637 1/20 0.37
PLA2G10 O15496 1/20 0.35
MGAM O43451 1/20 0.35
PLA2G2A P14555 1/20 0.35
PLA2G5 P39877 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29965948 0.75 TP53 (0.59) TNKSTNKS2PARP1ADORA3SLC6A3
SCHEMBL28895087 0.74 PARP1 (0.46) PDE5APDE9APARP1TP53
SCHEMBL29965256 0.74 PARP1 (0.42) PDE5APDE9APARP1TP53PLA2G10
SCHEMBL3337877 0.72 PARP1 (0.51) PDE5APDE9APARP1ADORA3TP53
SCHEMBL28895268 0.70 ALDH1A1 (0.55) PARP1ADORA3
SCHEMBL29965925 0.70 ALDH1A1 (0.55) PARP1ADORA3
SCHEMBL29965714 0.69 PARP1 (0.51) PARP1
SCHEMBL3583998 0.65 PDE9A (0.57) PDE5APDE9ATNKSTNKS2PARP1
SCHEMBL3592998 0.63 TNKS (0.45) PDE5APDE9ATNKSTNKS2PARP1
SCHEMBL3496118 0.62 PDE5A (1.00) PDE5APDE9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115368362-A Quinoxalinone derivatives as BTK inhibitors and application thereof 华东理工大学 2022-11-22 CN disclosed