SCHEMBL29967987

SCHEMBL29967987

Nc1nn(C(=O)CCC(=O)O)c2cccc(-c3ccc(C4=CCCCC4)cc3)c12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HDAC1 Q13547 6/20 0.36
HDAC2 Q92769 6/20 0.36
HDAC3 O15379 4/20 0.36
KDR P35968 5/20 0.36
FLT3 P36888 3/20 0.36
ACMSD Q8TDX5 1/20 0.35
PTGER1 P34995 1/20 0.35
PTGS2 P35354 1/20 0.34
TBK1 Q9UHD2 2/20 0.34
IKBKE Q14164 1/20 0.34
PAX8 Q06710 1/20 0.33
LCK P06239 1/20 0.33
CSF1R P07333 1/20 0.33
KIT P10721 1/20 0.33
FLT1 P17948 1/20 0.33
FLT4 P35916 1/20 0.33
ATR Q13535 1/20 0.33
GCGR P47871 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29967871 0.80 BTK (0.38) HDAC1HDAC2HDAC3KDRFLT3
SCHEMBL29967525 0.80 GCGR (0.35) MEN1KMT2AACMSDPTGER1GCGR
SCHEMBL29967807 0.78 KDR (0.50) HDAC1HDAC2HDAC3KDRFLT3
SCHEMBL29968057 0.77 PTGDR2 (0.36) MEN1KMT2A
SCHEMBL29967767 0.68 FABP4 (0.37) MEN1KMT2AACMSDPTGS2
SCHEMBL21386468 0.68 KDR (0.37) HDAC1HDAC2HDAC3KDRFLT3
SCHEMBL29967688 0.67 CNR2 (0.38) ACMSDPTGS2
SCHEMBL29967824 0.66 KDM4E (0.49) MEN1KMT2APTGS2
SCHEMBL29968082 0.65 KDR (0.63) KDRFLT3LCKCSF1RKIT
SCHEMBL11857930 0.65 ACMSD (0.54) HDAC1HDAC2HDAC3ACMSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed