SCHEMBL29967871

SCHEMBL29967871

CC(C)(C)OC(=O)n1nc(N)c2c(-c3ccc(C4=CCCCC4)cc3)cccc21

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BTK Q06187 2/20 0.38
NR1H2 P55055 1/20 0.37
KDR P35968 3/20 0.36
FLT3 P36888 3/20 0.36
MAP2K4 P45985 1/20 0.36
PDK4 Q16654 1/20 0.36
HDAC1 Q13547 8/20 0.35
HDAC2 Q92769 8/20 0.35
HDAC3 O15379 3/20 0.35
PTGS2 P35354 1/20 0.35
SMARCA2 P51531 1/20 0.35
SMARCA4 P51532 1/20 0.35
PBRM1 Q86U86 1/20 0.35
LCK P06239 1/20 0.34
CSF1R P07333 1/20 0.34
KIT P10721 1/20 0.34
FLT1 P17948 1/20 0.34
FLT4 P35916 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL421224 0.84 KDR (0.41) NR1H2KDRFLT3MAP2K4SMARCA2
SCHEMBL29967811 0.82 MAP2K4 (0.44) NR1H2KDRFLT3MAP2K4SMARCA2
SCHEMBL28871230 0.82 MAP2K4 (0.44) NR1H2KDRFLT3MAP2K4SMARCA2
SCHEMBL29967987 0.80 MEN1 (0.37) KDRFLT3HDAC1HDAC2HDAC3
SCHEMBL29967807 0.75 KDR (0.50) KDRFLT3HDAC1HDAC2HDAC3
SCHEMBL186237 0.72 MAP2K4 (0.41) NR1H2MAP2K4SMARCA2SMARCA4PBRM1
SCHEMBL185524 0.70 MAP2K4 (0.39) NR1H2MAP2K4SMARCA2SMARCA4PBRM1
SCHEMBL3668968 0.70 MAP2K4 (0.44) NR1H2MAP2K4SMARCA2SMARCA4PBRM1
SCHEMBL31319772 0.69 KDR (0.57) KDRFLT1
SCHEMBL1347906 0.68 KDR (0.59) KDRFLT3LCKCSF1RKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed