SCHEMBL29973807

SCHEMBL29973807

CN(C)C(=O)Cn1cc2cc(Br)ccc2n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.43
HDAC8 Q9BY41 1/20 0.41
IRAK4 Q9NWZ3 6/20 0.40
POLB P06746 1/20 0.40
CCNC P24863 2/20 0.39
CDK8 P49336 2/20 0.39
NCEH1 Q6PIU2 1/20 0.38
LMNA P02545 1/20 0.37
HDAC6 Q9UBN7 1/20 0.36
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
NPC1 O15118 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
RAB9A P51151 1/20 0.35
DYRK1A Q13627 1/20 0.35
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23320737 0.82 HDAC8 (0.47) S1PR1HDAC8IRAK4HDAC6
SCHEMBL22452466 0.81 S1PR1 (0.44) S1PR1HDAC8IRAK4CDK8LMNA
SCHEMBL15447288 0.81 CASP3 (0.49) S1PR1HDAC8IRAK4HDAC6NPC1
SCHEMBL30188651 0.77 HDAC8 (0.39) S1PR1HDAC8IRAK4HDAC6NPC1
SCHEMBL1637329 0.76 HDAC8 (0.39) HDAC8POLBHDAC6NPC1CYP1A2
SCHEMBL21411441 0.75 IRAK4 (0.38) HDAC8IRAK4
SCHEMBL28877889 0.75 S1PR1 (0.39) S1PR1IRAK4CCNCCDK8
SCHEMBL13332262 0.74 ALDH1A1 (0.43) S1PR1HDAC8POLBCDK8LMNA
SCHEMBL29209083 0.73 HDAC8 (0.42) S1PR1HDAC8IRAK4LMNAHDAC6
SCHEMBL31394603 0.73 HDAC8 (0.38) HDAC8IRAK4CCNCCDK8LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022206730-A1 PYRIMIDOPYRAZINE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-06 WO disclosed
CN-115141202-A Pyrimidopyrazinone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-04 CN disclosed