SCHEMBL29977870

SCHEMBL29977870

O=C(Nc1ccc(F)cc1F)N1CCc2sc(-c3noc(C(F)(F)F)n3)cc2C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.45
TAS1R1 Q7RTX1 1/20 0.45
TAS1R2 Q8TE23 1/20 0.45
ALDH1A1 P00352 2/20 0.39
PKM P14618 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HDAC6 Q9UBN7 5/20 0.39
HDAC8 Q9BY41 2/20 0.39
HDAC1 Q13547 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
MAPT P10636 2/20 0.38
POLB P06746 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
HDAC4 P56524 2/20 0.37
HDAC2 Q92769 1/20 0.37
OPRM1 P35372 1/20 0.37
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29977903 0.93 TAS1R3 (0.43) TAS1R3TAS1R1TAS1R2ALDH1A1PKM
SCHEMBL29978892 0.92 RAB9A (0.41) TAS1R3TAS1R1TAS1R2HDAC6HDAC8
SCHEMBL29978083 0.89 NPC1 (0.47) HDAC6HDAC8HDAC1SMN1; SMN2MAPT
SCHEMBL29978477 0.87 NPC1 (0.42) TAS1R3TAS1R1TAS1R2KDM4EHDAC6
SCHEMBL29978228 0.86 CYP3A4 (0.44) HDAC6HDAC8HDAC1SMN1; SMN2MAPT
SCHEMBL29978312 0.86 HDAC6 (0.39) HDAC6HDAC8HDAC1SMN1; SMN2MAPT
SCHEMBL29978715 0.86 MAPT (0.42) ALDH1A1PKMHDAC6MAPTPOLB
SCHEMBL29978177 0.85 MEN1 (0.41) ALDH1A1KDM4EHDAC6HDAC8HDAC1
SCHEMBL29978771 0.85 POLB (0.46) TAS1R3TAS1R1TAS1R2HDAC6HDAC8
SCHEMBL29978205 0.84 HDAC4 (0.47) HDAC6HDAC8HDAC1SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO claimed
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO disclosed