SCHEMBL29978477

SCHEMBL29978477

O=C(Nc1cccc(F)c1F)N1CCc2sc(-c3noc(C(F)(F)F)n3)cc2C1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
HDAC6 Q9UBN7 7/20 0.40
HDAC8 Q9BY41 4/20 0.40
HDAC1 Q13547 3/20 0.40
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
TAS1R2 Q8TE23 1/20 0.39
CSNK1D P48730 1/20 0.37
CSNK1E P49674 1/20 0.37
KDM4E B2RXH2 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
HDAC4 P56524 6/20 0.36
HDAC2 Q92769 1/20 0.36
GPR142 Q7Z601 2/20 0.35
P2RY1 P47900 2/20 0.35
BACE1 P56817 1/20 0.35
NTRK1 P04629 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29978771 0.87 POLB (0.46) NPC1RAB9AHDAC6HDAC8HDAC1
SCHEMBL29977870 0.87 TAS1R3 (0.45) NPC1RAB9AHDAC6HDAC8HDAC1
SCHEMBL29978721 0.87 DGAT1 (0.45) NPC1RAB9AHDAC6HDAC8HDAC1
SCHEMBL29978296 0.86 NPC1 (0.50) NPC1RAB9AHDAC6HDAC8HDAC1
SCHEMBL29978228 0.86 CYP3A4 (0.44) NPC1RAB9AHDAC6HDAC8HDAC1
SCHEMBL29978205 0.85 HDAC4 (0.47) NPC1RAB9AHDAC6HDAC8HDAC1
SCHEMBL29978115 0.85 DGAT1 (0.40) NPC1RAB9AHDAC6HDAC8HDAC1
SCHEMBL29978083 0.84 NPC1 (0.47) NPC1RAB9AHDAC6HDAC8HDAC1
SCHEMBL29978258 0.84 NPC1 (0.52) NPC1RAB9AHDAC6HDAC8HDAC1
SCHEMBL29978312 0.84 HDAC6 (0.39) NPC1RAB9AHDAC6HDAC8HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO claimed
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO disclosed