SCHEMBL29978115

SCHEMBL29978115

O=C(Nc1c(Cl)cccc1Cl)N1CCc2sc(-c3noc(C(F)(F)F)n3)cc2C1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 5/20 0.40
HDAC6 Q9UBN7 8/20 0.38
HDAC4 P56524 4/20 0.38
HDAC8 Q9BY41 4/20 0.38
HDAC1 Q13547 4/20 0.38
HDAC2 Q92769 1/20 0.38
NPC1 O15118 1/20 0.37
CASP3 P42574 1/20 0.37
RAB9A P51151 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
TAS1R3 Q7RTX0 2/20 0.37
TAS1R1 Q7RTX1 2/20 0.37
TAS1R2 Q8TE23 2/20 0.37
TRPM8 Q7Z2W7 1/20 0.36
CGAS Q8N884 1/20 0.36
HDAC5 Q9UQL6 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29978721 0.95 DGAT1 (0.45) DGAT1HDAC6HDAC4HDAC8HDAC1
SCHEMBL29977864 0.93 DGAT1 (0.40) DGAT1HDAC6HDAC4HDAC8HDAC1
SCHEMBL29978771 0.91 POLB (0.46) DGAT1HDAC6HDAC4HDAC8HDAC1
SCHEMBL29978258 0.89 NPC1 (0.52) HDAC6HDAC4HDAC8HDAC1NPC1
SCHEMBL29978321 0.88 MEN1 (0.47) HDAC6HDAC4HDAC8HDAC2NPC1
SCHEMBL29977980 0.87 HDAC4 (0.39) HDAC6HDAC4HDAC8HDAC1HDAC2
SCHEMBL29977881 0.87 MAPT (0.39) HDAC6HDAC4HDAC8HDAC1HDAC2
SCHEMBL29978205 0.87 HDAC4 (0.47) HDAC6HDAC4HDAC8HDAC1HDAC2
SCHEMBL29978361 0.86 TP53 (0.39) HDAC6HDAC4HDAC8HDAC1HDAC2
SCHEMBL29978228 0.85 CYP3A4 (0.44) HDAC6HDAC4HDAC8HDAC1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO claimed
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO disclosed