SCHEMBL29978664

SCHEMBL29978664

CN1CCN(c2ccc(-c3nccc(CO)n3)cn2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
CYP1A2 P05177 3/20 0.52
HSD17B10 Q99714 3/20 0.52
CYP3A4 P08684 2/20 0.52
CLK4 Q9HAZ1 2/20 0.52
CYP2D6 P10635 2/20 0.52
TSHR P16473 1/20 0.52
USP2 O75604 1/20 0.49
CASP1 P29466 1/20 0.49
CASP7 P55210 1/20 0.49
ALOX15 P16050 1/20 0.47
FYN P06241 4/20 0.45
TDO2 P48775 1/20 0.43
TNKS O95271 1/20 0.42
ZAP70 P43403 1/20 0.42
HRH4 Q9H3N8 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
HDAC1 Q13547 1/20 0.42
TLR9 Q9NR96 1/20 0.41
HTR3A P46098 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29979116 0.86 CNR2 (0.51) ALDH1A1HSD17B10ALOX15
SCHEMBL16815333 0.74 ACHE (0.50) HRH4HRH3HTR3ASORD
SCHEMBL11988947 0.72 SMO (0.52) FYNTDO2HRH4HRH3HTR3A
SCHEMBL24007658 0.72 CLK2 (0.43)
SCHEMBL30274584 0.72 CLK2 (0.43)
SCHEMBL31587676 0.71 TRPV3 (0.43) CYP3A4CLK4HDAC1RAB9ADYRK1A
SCHEMBL20420302 0.70 FYN (0.45) ALDH1A1CYP1A2HSD17B10CYP3A4CLK4
SCHEMBL29883568 0.70 HRH4 (0.62) FYNTNKSZAP70HRH4HRH3
SCHEMBL25082177 0.70 CNR2 (0.52) ALDH1A1CYP1A2HSD17B10CLK4TSHR
SCHEMBL29979194 0.70 GFER (0.49) ALDH1A1CYP1A2HSD17B10TSHRUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022216945-A1 MACROCYCLIC MCL1 INHIBITORS AND USES THEREOF CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-10-13 WO disclosed