SCHEMBL299826

SCHEMBL299826

C=CC(OC(=O)C(=C)C)Oc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.42
MTNR1A P48039 4/20 0.39
MTNR1B P49286 4/20 0.39
GAA P10253 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
PKM P14618 1/20 0.35
CYP2C19 P33261 1/20 0.35
HPGD P15428 2/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
KMT2A Q03164 1/20 0.33
THRB P10828 1/20 0.33
PPARG P37231 1/20 0.33
PPARA Q07869 1/20 0.33
TGM2 P21980 1/20 0.33
KDM4E B2RXH2 1/20 0.33
LTB4R Q15722 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8627211 0.87 KMT2A (0.49) ELANEPKMHPGDALDH1A1TP53
SCHEMBL1419286 0.85 MTNR1A (0.41) ELANEMTNR1AMTNR1BGAACYP1A2
SCHEMBL2861044 0.79 POLB (0.40) ELANEALDH1A1
SCHEMBL9662590 0.79 PARP10 (0.41) MTNR1AMTNR1BGAACYP1A2CYP2C9
SCHEMBL17351289 0.79 ELANE (0.45) ELANEMTNR1AMTNR1BGAACYP1A2
SCHEMBL21370 0.79 MTNR1A (0.45) ELANEMTNR1AMTNR1BGAACYP1A2
SCHEMBL299999 0.79 THRB (0.46) MTNR1AMTNR1BGAACYP1A2CYP2C9
SCHEMBL9461692 0.78 TSHR (0.44) ELANEMTNR1AMTNR1BGAACYP1A2
SCHEMBL9994926 0.77 THRB (0.39) ELANEMTNR1AMTNR1BGAACYP1A2
SCHEMBL10875073 0.77 LMNA (0.43) ELANEALDH1A1MEN1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 109 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3235852-A1 PHOTOACTIVE POLYMER MATERIALS Rolic AG (CH) 2017-10-25 EP claimed
EP-2655478-B1 PHOTOACTIVE POLYMER MATERIALS ROLIC AG (CH) 2017-06-14 EP claimed
EP-2655478-A1 PHOTOACTIVE POLYMER MATERIALS Rolic AG (CH) 2013-10-30 EP claimed
US-20130281564-A1 PHOTOACTIVE POLYMER MATERIALS ROLIC AG (CH) 2013-10-24 US claimed
US-8500807-B2 Photochromic intraocular lens CARL ZEISS MEDITEC SAS (FR) 2013-08-06 US claimed
WO-2012085048-A1 PHOTOACTIVE POLYMER MATERIALS ROLIC AG (CH) 2012-06-28 WO claimed
EP-1834195-B9 PHOTOCHROMIC INTRAOCULAR LENS IOLTECHNOLOGIE PRODUCTION (FR) 2010-07-21 EP claimed
EP-1834195-B1 PHOTOCHROMIC INTRAOCULAR LENS IOLTECHNOLOGIE PRODUCTION (FR) 2010-03-17 EP claimed
US-20080200983-A1 Photochromic Intraocular Lens IOLTECHNOLOGIE-PRODUCTION (FR) 2008-08-21 US claimed
JP-2008526334-A 2008-07-24 JP claimed
WO-2000026698-B1 INTRAOCULAR LENSES MADE FROM POLYMERIC COMPOSITIONS ALLERGAN SALES INC (US) 2000-07-13 WO claimed
WO-2000026698-A1 INTRAOCULAR LENSES MADE FROM POLYMERIC COMPOSITIONS ALLERGAN SALES, INC. (US) 2000-05-11 WO claimed
US-6014488-A Coated optical fibers having strippable primary coatings and processes for making and using same HEXION INC. (FORMERLY KNOWN AS MOMENTIVE SPECIALTY CHEMICALS INC.) 2000-01-11 US claimed
EP-0895606-A1 COATED OPTICAL FIBERS HAVING A REDUCED CONTENT OF EXTRACTABLE AND VOLATILE MATERIAL BORDEN CHEMICAL, INC. (US) 1999-02-10 EP claimed
EP-0894277-A1 COATED OPTICAL FIBERS HAVING STRIPPABLE PRIMARY COATINGS AND PROCESSES FOR MAKING AND USING SAME BORDEN CHEMICAL, INC. (US) 1999-02-03 EP claimed
WO-1998033081-A1 COATED OPTICAL FIBERS HAVING STRIPPABLE PRIMARY COATINGS AND PROCESSES FOR MAKING AND USING SAME BORDEN CHEMICAL, INC. (US) 1998-07-30 WO claimed
WO-1998019189-A1 COATED OPTICAL FIBERS HAVING A REDUCED CONTENT OF EXTRACTABLE AND VOLATILE MATERIAL BORDEN CHEMICAL, INC. (US) 1998-05-07 WO claimed
US-5744514-A PROTECTIVE COATING COMPRISING A RADIATION-CURED MERCAPTO-TERMINATED URETHANE OLIGOMER, A (METH)ACRYLATED POLYURETHANE AND AN ACRYLATE DILUENT; HEAT AND SOLVENT RESISTANCE; HIGH TENSILE MODULUS BORDEN CHEMICAL, INC. (US) 1998-04-28 US claimed
US-5591562-A SOLDER RESISTS, EPOXY RESINS WITH POLYMERIZABLE UNSATURATION AND QUATERNARY AMMONIUM, SULFONIUM OR PHOSPHONIUM GROUPS SONY CORPORATION (JP) 1997-01-07 US claimed
US-4133942-A Polymeric carrier for a controlled synthesis of peptides and the method of its preparation CESKOSLOVENSKA AKADEMIE VED (CS) 1979-01-09 US claimed