SCHEMBL29995997

SCHEMBL29995997

COC(=O)c1cccnc1N1C=CC=CC1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.43
KDM4E B2RXH2 1/20 0.43
OPRK1 P41145 7/20 0.43
CNR2 P34972 1/20 0.43
HRH3 Q9Y5N1 1/20 0.42
MAP2K1 Q02750 1/20 0.41
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
PKM P14618 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29995230 0.83 MYC (0.50) TDP1KDM4EALDH1A1L3MBTL1
SCHEMBL29995315 0.82 PARP1 (0.42) TDP1KDM4EALDH1A1
SCHEMBL29995876 0.79 L3MBTL1 (0.46) TDP1KDM4ECNR2MAP2K1ALDH1A1
SCHEMBL29994976 0.78 MYC (0.51) KDM4EALDH1A1L3MBTL1
SCHEMBL30118900 0.74 L3MBTL1 (0.34) KDM4EALDH1A1L3MBTL1
SCHEMBL30397636 0.73 L3MBTL1 (0.62) OPRK1HRH3ALDH1A1L3MBTL1
SCHEMBL38658667 0.73 L3MBTL1 (0.62) OPRK1HRH3ALDH1A1L3MBTL1
SCHEMBL15714564 0.72 MYC (0.69) TDP1KDM4EMAP2K1ALDH1A1TP53
SCHEMBL31317231 0.71 OPRK1 (0.58) TDP1KDM4EOPRK1CNR2HRH3
SCHEMBL7238484 0.71 CHIA (0.66) KDM4EOPRK1HRH3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115335043-A PGDH inhibitors and methods of making and using 迈欧伏特治疗公司 2022-11-11 CN disclosed