SCHEMBL30002369

SCHEMBL30002369

Cc1c(F)ccc2ncsc12

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.36
TGFBR1 P36897 2/20 0.35
ALDH1A1 P00352 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PKLR P30613 1/20 0.31
NPC1 O15118 4/20 0.31
RAB9A P51151 4/20 0.31
PFKFB3 Q16875 1/20 0.30
CDK1 P06493 1/20 0.30
CDK2 P24941 1/20 0.30
ABL1 P00519 1/20 0.30
KDM4E B2RXH2 1/20 0.30
HKDC1 Q2TB90 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8306186 0.79 ALDH1A1 (0.35) P2RX7ALDH1A1HSD17B10NPC1RAB9A
SCHEMBL659694 0.76 ALDH1A1 (0.33) TGFBR1ALDH1A1HSD17B10NPC1RAB9A
SCHEMBL4075607 0.76 ALDH1A1 (0.33) P2RX7ALDH1A1HSD17B10NPC1RAB9A
SCHEMBL3185104 0.76 DYRK1A (0.35) P2RX7ALDH1A1HSD17B10NPC1RAB9A
SCHEMBL12121766 0.76 ABL1 (0.34) P2RX7TGFBR1ALDH1A1HSD17B10NPC1
SCHEMBL18876099 0.76 P2RX7 (0.34) P2RX7ALDH1A1HSD17B10NPC1RAB9A
SCHEMBL6068320 0.76 CCNE1 (0.37) P2RX7TGFBR1ALDH1A1HSD17B10PKLR
SCHEMBL2722669 0.75 ALDH1A1 (0.46) ALDH1A1HSD17B10NPC1RAB9ACDK1
SCHEMBL18876131 0.74 TGFBR1 (0.36) TGFBR1
SCHEMBL29324220 0.73 ADORA2A (0.33) P2RX7TGFBR1ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed