SCHEMBL30002392

SCHEMBL30002392

COc1cc(F)c([N+](=O)[O-])cc1OCc1cccc2nccnc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
GAA P10253 4/20 0.41
PKM P14618 1/20 0.41
ALDH1A1 P00352 7/20 0.40
LMNA P02545 5/20 0.40
MAPT P10636 4/20 0.40
PTGES O14684 2/20 0.40
HPGD P15428 2/20 0.40
POLB P06746 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
CHEK1 O14757 1/20 0.39
KDM4E B2RXH2 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892472 1.00 KMT2A (0.46) KMT2AMEN1GAAPKMALDH1A1
SCHEMBL30003288 0.88 GAA (0.40) KMT2AMEN1GAAPKMALDH1A1
SCHEMBL30001950 0.87 ALDH1A1 (0.52) KMT2AMEN1GAAPKMALDH1A1
SCHEMBL28892294 0.87 ALDH1A1 (0.52) KMT2AMEN1GAAPKMALDH1A1
SCHEMBL30003416 0.84 KMT2A (0.50) KMT2AMEN1GAAPKMALDH1A1
SCHEMBL28892412 0.84 KMT2A (0.50) KMT2AMEN1GAAPKMALDH1A1
SCHEMBL30002459 0.82 GAA (0.48) KMT2AMEN1GAAPKMALDH1A1
SCHEMBL30003319 0.81 GAA (0.40) KMT2AMEN1GAAPKMALDH1A1
SCHEMBL28892476 0.81 MEN1 (0.52) KMT2AMEN1GAAPKMALDH1A1
SCHEMBL30002031 0.81 DHFR (0.38) KMT2AMEN1GAAPKMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed