SCHEMBL30002459

SCHEMBL30002459

COc1cc(F)c([N+](=O)[O-])cc1NCc1cccc2nccnc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.48
PKM P14618 2/20 0.48
MEN1 O00255 6/20 0.44
KMT2A Q03164 6/20 0.44
MAPT P10636 10/20 0.43
HTT P42858 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ALDH1A1 P00352 7/20 0.42
MAPK1 P28482 3/20 0.42
KDM4E B2RXH2 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
POLB P06746 2/20 0.40
TP53 P04637 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
HPGD P15428 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892472 0.82 KMT2A (0.46) GAAPKMMEN1KMT2AMAPT
SCHEMBL30002392 0.82 KMT2A (0.46) GAAPKMMEN1KMT2AMAPT
SCHEMBL30002823 0.82 DHFR (0.43) GAAMEN1KMT2AMAPTHTT
SCHEMBL28892864 0.82 DHFR (0.43) GAAMEN1KMT2AMAPTHTT
SCHEMBL28892417 0.79 GAA (0.52) GAAPKMMEN1KMT2AMAPT
SCHEMBL30002395 0.78 GAA (0.47) GAAPKMMEN1KMT2AMAPT
SCHEMBL28892666 0.78 GAA (0.47) GAAPKMMEN1KMT2AMAPT
SCHEMBL28892688 0.76 CD274 (0.35) GAAMEN1KMT2AMAPTHTT
SCHEMBL2932177 0.72 GAA (0.45) GAAPKMMEN1KMT2AMAPT
SCHEMBL30002765 0.72 GAA (0.45) GAAPKMMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed