SCHEMBL30002519

SCHEMBL30002519

COc1cc(F)c(N)cc1OCc1cccc2ncsc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.37
DCPS Q96C86 2/20 0.37
KIT P10721 1/20 0.37
CSF1R P07333 3/20 0.36
KMT2A Q03164 2/20 0.36
CHRM1 P11229 1/20 0.35
PARP10 Q53GL7 2/20 0.33
KDR P35968 2/20 0.33
PKM P14618 1/20 0.33
PARP15 Q460N3 1/20 0.33
PARP14 Q460N5 1/20 0.33
CYP1A2 P05177 1/20 0.33
EPHA2 P29317 1/20 0.33
EPHB4 P54760 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29211328 1.00 DHFR (0.37) DHFRDCPSKITCSF1RKMT2A
SCHEMBL28892418 0.83 KIT (0.37) KITCSF1RKMT2AKDREPHA2
SCHEMBL30003338 0.83 KIT (0.37) KITCSF1RKMT2AKDREPHA2
SCHEMBL30003319 0.82 GAA (0.40) KMT2APKMCYP1A2MAPTMEN1
SCHEMBL28892714 0.82 GAA (0.40) KMT2APKMCYP1A2MAPTMEN1
SCHEMBL30002757 0.82 KIT (0.34) DHFRDCPSKITCSF1RKMT2A
SCHEMBL28892349 0.82 KIT (0.34) DHFRDCPSKITCSF1RKMT2A
SCHEMBL30002396 0.81 KIT (0.35) DHFRKITCSF1RKMT2AMAPT
SCHEMBL28892739 0.81 KIT (0.35) DHFRKITCSF1RKMT2AMAPT
SCHEMBL30002031 0.79 DHFR (0.38) DHFRDCPSKITCSF1RKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed