SCHEMBL30002570

SCHEMBL30002570

COc1cc(F)c([N+](=O)[O-])cc1OCc1cccc2ccc(C)nc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.52
KMT2A Q03164 4/20 0.52
ALDH1A1 P00352 3/20 0.45
PTGDR2 Q9Y5Y4 1/20 0.43
RELA Q04206 2/20 0.42
LMNA P02545 3/20 0.41
MAPT P10636 3/20 0.41
POLB P06746 2/20 0.41
HPGD P15428 1/20 0.41
GAA P10253 1/20 0.40
PKM P14618 1/20 0.40
NFKBIA P25963 1/20 0.40
PTGES O14684 1/20 0.40
ALOX5 P09917 1/20 0.39
RAB9A P51151 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892476 1.00 MEN1 (0.52) MEN1KMT2AALDH1A1PTGDR2RELA
SCHEMBL30002646 0.90 LMNA (0.41) MEN1KMT2AALDH1A1LMNAMAPT
SCHEMBL28892509 0.90 LMNA (0.41) MEN1KMT2AALDH1A1LMNAMAPT
SCHEMBL30001950 0.88 ALDH1A1 (0.52) MEN1KMT2AALDH1A1LMNAMAPT
SCHEMBL28892294 0.88 ALDH1A1 (0.52) MEN1KMT2AALDH1A1LMNAMAPT
SCHEMBL30002629 0.86 HTR1A (0.41) MEN1KMT2AALDH1A1RELALMNA
SCHEMBL28892764 0.84 HTR1A (0.41) MEN1KMT2AALDH1A1LMNAMAPT
SCHEMBL30002600 0.84 HTR1A (0.41) MEN1KMT2AALDH1A1LMNAMAPT
SCHEMBL30002023 0.82 GAA (0.39) MEN1KMT2AALDH1A1RELALMNA
SCHEMBL30002421 0.82 MEN1 (0.47) MEN1KMT2AALDH1A1PTGDR2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed