SCHEMBL30002604

SCHEMBL30002604

COc1cc(F)c(N)cc1OCc1ccc(Cl)c2scnc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.34
EPHA2 P29317 6/20 0.34
KDR P35968 6/20 0.34
EPHB4 P54760 6/20 0.34
KIT P10721 1/20 0.33
ERBB2 P04626 3/20 0.33
G6PD P11413 1/20 0.32
EGFR P00533 1/20 0.32
LMNA P02545 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CSF1R P07333 1/20 0.32
HDAC8 Q9BY41 2/20 0.31
GAA P10253 1/20 0.31
STING1 Q86WV6 1/20 0.31
FLT1 P17948 1/20 0.31
DYRK1A Q13627 1/20 0.30
NFKB1 P19838 1/20 0.30
RAB9A P51151 1/20 0.30
NFKB2 Q00653 1/20 0.30
RELA Q04206 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892360 1.00 NPC1 (0.34) NPC1EPHA2KDREPHB4KIT
SCHEMBL28892739 0.90 KIT (0.35) NPC1KITCSF1RGAARAB9A
SCHEMBL30002396 0.90 KIT (0.35) NPC1KITCSF1RGAARAB9A
SCHEMBL28892649 0.83 NPC1 (0.35) NPC1EPHA2KDREPHB4KIT
SCHEMBL30002017 0.83 NPC1 (0.35) NPC1EPHA2KDREPHB4KIT
SCHEMBL28959472 0.83 LMNA (0.38) NPC1LMNAGAARAB9ASMN1; SMN2
SCHEMBL30002416 0.83 LMNA (0.38) NPC1LMNAGAARAB9ASMN1; SMN2
SCHEMBL28892550 0.80 EPHA2 (0.37) NPC1EPHA2KDREPHB4KIT
SCHEMBL30002766 0.80 EPHA2 (0.37) NPC1EPHA2KDREPHB4KIT
SCHEMBL30002757 0.80 KIT (0.34) EPHA2KDREPHB4KITCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed