SCHEMBL30002765

SCHEMBL30002765

COc1cc(F)c([N+](=O)[O-])cc1NCc1c(OC)ccc(F)c1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.45
PKM P14618 1/20 0.45
MAPT P10636 9/20 0.44
KMT2A Q03164 7/20 0.44
ALDH1A1 P00352 6/20 0.44
MEN1 O00255 5/20 0.44
MAPK1 P28482 3/20 0.43
CRHBP P24387 3/20 0.43
CRHR2 Q13324 3/20 0.43
HTT P42858 4/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ABCB1 P08183 2/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2932177 1.00 GAA (0.45) GAAPKMMAPTKMT2AALDH1A1
SCHEMBL28892279 0.93 GAA (0.42) GAAPKMMAPTKMT2AALDH1A1
SCHEMBL28892445 0.91 GAA (0.41) GAAPKMMAPTKMT2AALDH1A1
SCHEMBL28892707 0.89 GAA (0.39) GAAPKMMAPTKMT2AALDH1A1
SCHEMBL28892141 0.79 HTR2A (0.37) GAAMAPTKMT2AALDH1A1MEN1
SCHEMBL30003307 0.78 GNRHR (0.42) GAAPKMMAPTKMT2AALDH1A1
SCHEMBL10300131 0.78 GNRHR (0.42) GAAPKMMAPTKMT2AALDH1A1
SCHEMBL28892882 0.76 ALDH1A1 (0.44) GAAPKMMAPTKMT2AALDH1A1
SCHEMBL30226326 0.76 ALDH1A1 (0.39) GAAPKMMAPTKMT2AALDH1A1
SCHEMBL28892793 0.75 RAB9A (0.38) GAAPKMMAPTKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed