SCHEMBL30003307

SCHEMBL30003307

COc1cc(F)c([N+](=O)[O-])cc1OCc1c(OC)ccc(F)c1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GNRHR P30968 1/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 2/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
LMNA P02545 5/20 0.41
ALDH1A1 P00352 12/20 0.40
MAPT P10636 7/20 0.40
MAPK1 P28482 3/20 0.40
KDM4E B2RXH2 2/20 0.40
ALOX15 P16050 1/20 0.40
PRKDC P78527 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GAA P10253 4/20 0.39
PKM P14618 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10300131 1.00 GNRHR (0.42) GNRHRMEN1KMT2ACYP3A4CYP2C19
SCHEMBL28892479 0.92 ALDH1A1 (0.41) GNRHRMEN1KMT2ACYP2C19NPC1
SCHEMBL28893037 0.91 KMT2A (0.40) GNRHRMEN1KMT2ACYP3A4CYP2C19
SCHEMBL28892160 0.89 GAA (0.42) GNRHRMEN1KMT2ACYP3A4CYP2C19
SCHEMBL3099715 0.89 LMNA (0.43) GNRHRMEN1KMT2ACYP3A4CYP2C19
SCHEMBL30001980 0.89 GNRHR (0.36) GNRHRCYP2C19LMNAALDH1A1GAA
SCHEMBL28892468 0.89 GNRHR (0.36) GNRHRCYP2C19LMNAALDH1A1GAA
SCHEMBL30002390 0.88 PDE4D (0.37) GNRHRMEN1KMT2ACYP3A4CYP2C19
SCHEMBL28892461 0.88 PDE4D (0.37) GNRHRMEN1KMT2ACYP3A4CYP2C19
SCHEMBL28892882 0.88 ALDH1A1 (0.44) MEN1KMT2ACYP3A4CYP2C19NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-116178389-A Preparation method of linagoli 浙江科聚生物医药有限公司 2023-05-30 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed