SCHEMBL30002838

SCHEMBL30002838

COc1cc(F)c(N)cc1NCc1cccc2cccnc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 10/20 0.55
KMT2A Q03164 10/20 0.55
MAPT P10636 4/20 0.55
ALDH1A1 P00352 4/20 0.55
HPGD P15428 3/20 0.55
PTBP1 P26599 1/20 0.55
HTT P42858 1/20 0.55
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
HTR2B P41595 1/20 0.48
ADORA2A P29274 3/20 0.46
ADORA1 P30542 3/20 0.46
L3MBTL1 Q9Y468 4/20 0.45
KDM4E B2RXH2 2/20 0.45
BLM P54132 2/20 0.44
NSD2 O96028 1/20 0.44
GAA P10253 1/20 0.42
RECQL P46063 1/20 0.42
LMNA P02545 3/20 0.42
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892277 1.00 MEN1 (0.55) MEN1KMT2AMAPTALDH1A1HPGD
SCHEMBL28892864 0.87 DHFR (0.43) MEN1KMT2AMAPTALDH1A1HPGD
SCHEMBL30002823 0.87 DHFR (0.43) MEN1KMT2AMAPTALDH1A1HPGD
SCHEMBL28892414 0.81 L3MBTL1 (0.48) MEN1KMT2AMAPTALDH1A1HPGD
SCHEMBL17208267 0.72 HDAC6 (0.52) MEN1KMT2AMAPTALDH1A1HPGD
SCHEMBL30003250 0.70 NSD2 (0.41) MEN1KMT2AMAPTALDH1A1NSD2
SCHEMBL28892537 0.70 NSD2 (0.41) MEN1KMT2AMAPTALDH1A1NSD2
SCHEMBL5118383 0.70 HDAC6 (0.50) MEN1KMT2AMAPTALDH1A1HPGD
SCHEMBL12748203 0.70 HDAC6 (0.60) MEN1KMT2AMAPTALDH1A1HPGD
SCHEMBL28892141 0.69 HTR2A (0.37) MEN1KMT2AMAPTALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed