SCHEMBL30002823

SCHEMBL30002823

COc1cc(F)c(N)cc1NCc1cccc2nccnc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.43
ALDH1A1 P00352 6/20 0.42
MAPT P10636 6/20 0.42
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
HPGD P15428 3/20 0.42
HTT P42858 2/20 0.42
PTBP1 P26599 1/20 0.42
L3MBTL1 Q9Y468 3/20 0.41
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
KDM4E B2RXH2 5/20 0.40
GAA P10253 4/20 0.40
LMNA P02545 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
POLB P06746 1/20 0.39
TSHR P16473 1/20 0.39
CRHBP P24387 1/20 0.39
MAPK1 P28482 1/20 0.39
CRHR2 Q13324 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892864 1.00 DHFR (0.43) DHFRALDH1A1MAPTKMT2AMEN1
SCHEMBL30002838 0.87 MEN1 (0.55) DHFRALDH1A1MAPTKMT2AMEN1
SCHEMBL28892277 0.87 MEN1 (0.55) DHFRALDH1A1MAPTKMT2AMEN1
SCHEMBL30002459 0.82 GAA (0.48) ALDH1A1MAPTKMT2AMEN1HPGD
SCHEMBL30002031 0.81 DHFR (0.38) DHFRMAPTKMT2AMEN1ADORA2A
SCHEMBL28892688 0.80 CD274 (0.35) DHFRALDH1A1MAPTKMT2AMEN1
SCHEMBL28892414 0.77 L3MBTL1 (0.48) DHFRALDH1A1MAPTKMT2AMEN1
SCHEMBL28892141 0.69 HTR2A (0.37) ALDH1A1MAPTKMT2AMEN1HPGD
SCHEMBL28892399 0.68 KIT (0.39) MAPTKMT2AMEN1GAATDP1
SCHEMBL622763 0.64 NQO2 (0.55) ALDH1A1MAPTKMT2AMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed