SCHEMBL30003147

SCHEMBL30003147

CON(C)C(=O)c1ccc(=O)n(COCC[Si](C)(C)C)n1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.34
NPC1 O15118 1/20 0.33
POLB P06746 2/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
KDM4E B2RXH2 3/20 0.32
ALDH1A1 P00352 1/20 0.32
HSD17B10 Q99714 1/20 0.32
PTGS1 P23219 1/20 0.32
DGAT1 O75907 3/20 0.32
MEN1 O00255 1/20 0.31
MAPT P10636 2/20 0.31
LMNA P02545 1/20 0.31
SAE1 Q9UBE0 1/20 0.31
UBA2 Q9UBT2 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
USP2 O75604 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24724344 0.83 KMT2A (0.38) KMT2ANPC1POLBKDM4EALDH1A1
SCHEMBL22393670 0.82 NPC1 (0.37) KMT2ANPC1POLBKDM4EALDH1A1
SCHEMBL30827496 0.82 NPC1 (0.37) KMT2ANPC1POLBKDM4EALDH1A1
SCHEMBL24724720 0.74 NPC1 (0.38) NPC1DGAT1
SCHEMBL26733973 0.74 DGAT1 (0.35) NPC1DGAT1
SCHEMBL29109010 0.72 KDM4E (0.34) KMT2ANPC1POLBKDM4EALDH1A1
SCHEMBL24667775 0.72 DGAT1 (0.40) KMT2ANPC1POLBKDM4EALDH1A1
SCHEMBL31728764 0.72 ALDH1A1 (0.43) KMT2ANPC1POLBKDM4EALDH1A1
SCHEMBL3594665 0.72 HPGD (0.39) KMT2ANPC1POLBKDM4EALDH1A1
SCHEMBL24724337 0.72 F2RL1 (0.36) KMT2ANPC1POLBKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240287070-A1 FUSED HETEROCYCLIC DERIVATIVES JOHNSON & JOHNSON (CHINA) INVESTMENT LTD. (CN) 2024-08-29 US disclosed
EP-4347590-A1 FUSED HETEROCYCLIC DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2024-04-10 EP disclosed
WO-2022253259-A1 FUSED HETEROCYCLIC DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2022-12-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240287070-A1 FUSED HETEROCYCLIC DERIVATIVES HAVCR2, HCCS, GOT2 KMT2A 3953/4885NPC1 95/4885POLB 587/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.