SCHEMBL30003246

SCHEMBL30003246

COc1cc(F)c([N+](=O)[O-])cc1OCc1cccc2ncncc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.40
PKM P14618 1/20 0.40
ABCG2 Q9UNQ0 2/20 0.39
HTR1A P08908 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
ALDH1A1 P00352 5/20 0.38
LMNA P02545 3/20 0.38
PTGES O14684 2/20 0.38
KMT2A Q03164 3/20 0.37
ACHE P22303 1/20 0.37
BACE1 P56817 1/20 0.37
EGFR P00533 1/20 0.37
CHEK1 O14757 1/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892628 1.00 GAA (0.40) GAAPKMABCG2HTR1AADRA1D
SCHEMBL28893045 0.85 SCN1A (0.46) GAAPKMHTR1AADRA1DADRA1A
SCHEMBL30002055 0.85 SCN1A (0.46) GAAPKMHTR1AADRA1DADRA1A
SCHEMBL30002926 0.82 KIT (0.41) PKMHTR1AALDH1A1KMT2AEGFR
SCHEMBL30003288 0.82 GAA (0.40) GAAPKMABCG2HTR1AADRA1D
SCHEMBL28892472 0.81 KMT2A (0.46) GAAPKMHTR1AADRA1DADRA1A
SCHEMBL30002392 0.81 KMT2A (0.46) GAAPKMHTR1AADRA1DADRA1A
SCHEMBL28892812 0.80 CHEK1 (0.41) GAAPKMALDH1A1LMNAKMT2A
SCHEMBL28892714 0.80 GAA (0.40) GAAPKMABCG2HTR1AADRA1D
SCHEMBL30003319 0.80 GAA (0.40) GAAPKMABCG2HTR1AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed