SCHEMBL30002926

SCHEMBL30002926

COc1cc(F)c(N)cc1OCc1cccc2ncncc12

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.41
KMT2A Q03164 1/20 0.40
DHFR P00374 3/20 0.37
DCPS Q96C86 2/20 0.37
EGFR P00533 2/20 0.36
CSF1R P07333 2/20 0.36
ALDH1A1 P00352 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
KDR P35968 4/20 0.36
EPHA2 P29317 2/20 0.36
HTR1A P08908 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
ERBB2 P04626 1/20 0.36
PKM P14618 1/20 0.35
FLT1 P17948 1/20 0.35
EPHB4 P54760 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892526 0.83 SCN1A (0.47)
SCHEMBL30002548 0.83 SCN1A (0.47)
SCHEMBL30003246 0.82 GAA (0.40) KMT2AEGFRALDH1A1HTR1APKM
SCHEMBL28892628 0.82 GAA (0.40) KMT2AEGFRALDH1A1HTR1APKM
SCHEMBL30002031 0.79 DHFR (0.38) KITKMT2ADHFRDCPSCSF1R
SCHEMBL28892213 0.78 KIT (0.37) KITKMT2AEGFRCSF1RKDR
SCHEMBL30002637 0.78 KIT (0.37) KITKMT2AEGFRCSF1RKDR
SCHEMBL30002519 0.77 DHFR (0.37) KITKMT2ADHFRDCPSCSF1R
SCHEMBL29211328 0.77 DHFR (0.37) KITKMT2ADHFRDCPSCSF1R
SCHEMBL30002665 0.76 SCN1A (0.37) KITKDREPHA2ERBB2FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed