SCHEMBL30005099

SCHEMBL30005099

CC1(C)OB(c2cccc3c2CCC(=O)N3)OC1(C)C

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
MAPK13 O15264 1/20 0.40
MAPK12 P53778 1/20 0.40
MAPK11 Q15759 1/20 0.40
MAPK14 Q16539 1/20 0.40
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
HTR1A P08908 1/20 0.36
OPRK1 P41145 1/20 0.36
MAPT P10636 1/20 0.35
JAK2 O60674 1/20 0.33
BTK Q06187 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22120124 1.00 NPC1 (0.40) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL29460881 0.87 DRD2 (0.41) HTR1AOPRK1
SCHEMBL1016712 0.87 DRD2 (0.41) HTR1AOPRK1
SCHEMBL31161182 0.79 NOTUM (0.34)
SCHEMBL15956758 0.79 NOTUM (0.34)
SCHEMBL17645720 0.78 JAK2 (0.32) JAK2BTK
SCHEMBL20595135 0.77 KDM1A (0.33)
SCHEMBL18342173 0.77 P2RX7 (0.35) HTR1AJAK2BTK
SCHEMBL31707905 0.76 ALDH1A1 (0.37) JAK2BTK
SCHEMBL508291 0.76 ALDH1A1 (0.37) JAK2BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4090660-A1 QUINOXALINE DERIVATIVES Grünenthal GmbH (DE) 2022-11-23 EP disclosed