SCHEMBL30006017

SCHEMBL30006017

NC(=O)Cc1ccc2cc[nH]c2c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 3/20 0.53
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 2/20 0.50
ENPP2 Q13822 2/20 0.50
HPGD P15428 1/20 0.50
HSD17B10 Q99714 1/20 0.50
TYR P14679 1/20 0.47
BACE1 P56817 4/20 0.46
CA2 P00918 1/20 0.44
CYP2A6 P11509 1/20 0.43
FAAH O00519 1/20 0.43
AHR P35869 2/20 0.43
CMA1 P23946 1/20 0.43
CACNA1G O43497 1/20 0.43
CACNA1H O95180 1/20 0.43
CACNA1I Q9P0X4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1607899 1.00 NLRP3 (0.53) NLRP3KDM4EALDH1A1ENPP2HPGD
SCHEMBL30006673 0.86 HDAC1 (0.54) KDM4EALDH1A1ENPP2CA2CYP2A6
SCHEMBL9225433 0.86 HDAC1 (0.54) KDM4EALDH1A1ENPP2CA2CYP2A6
SCHEMBL29627552 0.84 KDM4E (0.56) NLRP3KDM4EALDH1A1ENPP2HPGD
SCHEMBL3105331 0.84 KDM4E (0.56) NLRP3KDM4EALDH1A1ENPP2HPGD
SCHEMBL21274689 0.83 BACE1 (0.50) NLRP3KDM4EALDH1A1ENPP2HPGD
Water SCHEMBL8810335 0.83 KDM4E (0.54) NLRP3KDM4EALDH1A1ENPP2HPGD
SCHEMBL10645020 0.79 NLRP3 (0.60) NLRP3KDM4EALDH1A1ENPP2HPGD
SCHEMBL6675330 0.79 NLRP3 (0.64) NLRP3KDM4EALDH1A1ENPP2HPGD
SCHEMBL11976503 0.79 NLRP3 (0.53) NLRP3KDM4EALDH1A1ENPP2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4103278-A1 SMALL MOLECULE STING ANTAGONISTS Curadev Pharma Pvt. Ltd. (IN) 2022-12-21 EP claimed
EP-4337642-A1 ETHACRYNIC ACID DERIVATIVES AS INHIBITORS OF MPRO PROTEASE AND SARS-COV-2 REPLICATION Universite Euro-Mediterraneenne de Fes (MA) 2024-03-20 EP disclosed
CN-116554050-A Amide phenol derivative and application thereof 四川大学 2023-08-08 CN disclosed
EP-4103278-A1 SMALL MOLECULE STING ANTAGONISTS Curadev Pharma Pvt. Ltd. (IN) 2022-12-21 EP disclosed
CN-115427044-A Pyrrolopyrimidines as complement inhibitors 拜奥克里斯特制药公司 2022-12-02 CN disclosed
WO-2022240277-A1 ETHACRYNIC ACID DERIVATIVES AS INHIBITORS OF MPRO PROTEASE AND SARS-COV-2 REPLICATION UNIVERSITE EURO-MEDITERRANEENNE DE FES (MA) 2022-11-17 WO disclosed