SCHEMBL30006842

SCHEMBL30006842

COc1cccc(Cc2cccnc2C(N)=O)c1OC

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.45
KDM4E B2RXH2 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
NPC1 O15118 2/20 0.43
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA14 Q9ULX7 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
PLAU P00749 1/20 0.40
POLB P06746 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HIF1A Q16665 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30006783 0.88 TDP1 (0.49) RAB9AKDM4ENPC1TDP1TP53
SCHEMBL28001171 0.81 KDM4E (0.50) KDM4EL3MBTL1MAPTALDH1A1
SCHEMBL29503858 0.78 PLAU (0.53) RAB9AL3MBTL1NPC1CA12CA1
SCHEMBL1101140 0.78 PLAU (0.53) RAB9AL3MBTL1NPC1CA12CA1
SCHEMBL3306584 0.76 SMN1; SMN2 (0.54) RAB9AKDM4EL3MBTL1CA12CA1
SCHEMBL29056033 0.76 GRM2 (0.47) RAB9AKDM4ENPC1CA1CA2
SCHEMBL5250683 0.75 RAB9A (0.42) RAB9AKDM4EROCK2ROCK1CA12
SCHEMBL30006624 0.75 NR3C2 (0.42) KDM4EMAPTPLAU
SCHEMBL1503239 0.74 KDM4E (0.45) RAB9AKDM4EL3MBTL1NPC1TDP1
SCHEMBL8092420 0.74 KMT2A (0.54) KDM4ENPC1ROCK2ROCK1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111808023-B Method for preparing 3-aryl isoquinoline derivative 四川大学 2022-10-21 CN disclosed