SCHEMBL5250683

SCHEMBL5250683

COc1cccc(Cc2nc(O)c(O)c(C(N)=O)n2)c1OC

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.42
KMT2A Q03164 4/20 0.40
IKBKB O14920 1/20 0.39
NR3C2 P08235 1/20 0.39
MAOB P27338 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA14 Q9ULX7 1/20 0.38
MEN1 O00255 2/20 0.38
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
HPGD P15428 1/20 0.38
ALDH1A1 P00352 3/20 0.37
HIF1A Q16665 1/20 0.37
IDO1 P14902 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5119931 0.76 KDM4E (0.49) RAB9AKMT2AMAOBMEN1ROCK2
SCHEMBL5116129 0.76 MAOB (0.48) KMT2AMAOBMEN1ROCK2ROCK1
SCHEMBL30006842 0.75 RAB9A (0.45) RAB9AKMT2ACA12CA1CA2
SCHEMBL5118706 0.74 MAOB (0.48) RAB9AKMT2AMAOBMEN1ROCK2
SCHEMBL13729249 0.73 HTR6 (0.50) ALDH1A1IDO1LMNAKDM4E
SCHEMBL5121466 0.73 TDP1 (0.49) KMT2AMAOBROCK2ROCK1HPGD
SCHEMBL5128409 0.72 MAOB (0.48) KMT2AMAOBROCK2ROCK1HPGD
SCHEMBL5119117 0.72 MAOB (0.48) KMT2AMAOBMEN1ROCK2ROCK1
SCHEMBL5123346 0.71 HPGD (0.52) RAB9AKMT2AMAOBMEN1HPGD
SCHEMBL15458842 0.71 EGLN1 (0.47) RAB9AKMT2AMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441734-B1 DIHYDROXYPYRIMIDINE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE ANGELETTI P IST RICHERCHE BIO (IT) 2007-02-28 EP disclosed