SCHEMBL30007360

SCHEMBL30007360

COC(=O)c1c[nH]c2ncc(-c3ccc(S(C)(=O)=O)cc3)cc12

nearest known ligand 0.72

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AXL P30530 6/20 0.72
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
CAMKK2 Q96RR4 3/20 0.53
SGK1 O00141 1/20 0.53
AAK1 Q2M2I8 1/20 0.49
MAP2K1 Q02750 1/20 0.49
NR4A2 P43354 2/20 0.48
NEK1 Q96PY6 1/20 0.47
PIK3CA P42336 1/20 0.47
DYRK1A Q13627 2/20 0.47
CLK1 P49759 1/20 0.47
DYRK2 Q92630 1/20 0.47
DYRK1B Q9Y463 1/20 0.47
PAK1 Q13153 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL30007736 0.88 CAMKK2 (0.57) AXLCYP2C9CYP2C19CAMKK2SGK1
SCHEMBL30008314 0.87 AXL (0.67) AXLCYP2C9CYP2C19CAMKK2SGK1
SCHEMBL4119627 0.83 AXL (0.61) AXLCAMKK2SGK1AAK1
SCHEMBL4119636 0.82 MAP4K1 (0.67) AXLCYP2C19CAMKK2SGK1PAK1
SCHEMBL2891511 0.76 CYP2C19 (0.70) CYP2C9CYP2C19MAP2K1
SCHEMBL2891508 0.76 CYP2C19 (0.72) CYP2C9CYP2C19MAP2K1
Hydrochloric Acid SCHEMBL30007576 0.75 AXL (0.54) AXLCYP2C9CYP2C19CAMKK2SGK1
SCHEMBL16946570 0.75 CAMKK2 (0.51) AXLCYP2C9CYP2C19CAMKK2SGK1
SCHEMBL18238316 0.75 CAMKK2 (0.51) AXLCYP2C9CYP2C19CAMKK2SGK1
SCHEMBL7117672 0.75 CYP2C9 (0.53) CYP2C9CYP2C19CAMKK2SGK1AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022237922-A1 ANTITUMOR COMPOUNDS BASED ON NITROGEN HETEROCYCLES AND USE THEREOF AS MEDICAMENTS FAKULTNI NEMOCNICE HRADEC KRALOVE (CZ) 2022-11-17 WO disclosed