SCHEMBL30008314

SCHEMBL30008314

COC(=O)c1c[nH]c2ncc(-c3ccc(S(=O)(=O)C(C)C)cc3)cc12

nearest known ligand 0.67

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AXL P30530 6/20 0.67
CAMKK2 Q96RR4 2/20 0.50
SGK1 O00141 1/20 0.50
AAK1 Q2M2I8 1/20 0.47
MAP2K1 Q02750 1/20 0.46
NR4A2 P43354 2/20 0.46
NEK1 Q96PY6 4/20 0.45
PIK3CA P42336 1/20 0.45
DYRK1A Q13627 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL30007576 0.89 AXL (0.54) AXLCAMKK2SGK1AAK1PIK3CA
SCHEMBL30007360 0.87 AXL (0.72) AXLCAMKK2SGK1AAK1MAP2K1
SCHEMBL4119627 0.80 AXL (0.61) AXLCAMKK2SGK1AAK1
SCHEMBL30007677 0.80 AXL (0.50) AXLCAMKK2SGK1AAK1PIK3CA
SCHEMBL4119636 0.79 MAP4K1 (0.67) AXLCAMKK2SGK1CYP2C19
SCHEMBL30007734 0.79 MAPK8 (0.45) AXLCAMKK2PIK3CADYRK1A
SCHEMBL30007804 0.78 ALDH1A1 (0.46) AXLCYP2C9CYP2C19
SCHEMBL2887279 0.78 BRAF (0.59) MAP2K1CYP2C9CYP2C19
SCHEMBL2887275 0.77 CYP2C19 (0.59) MAP2K1CYP2C9CYP2C19
SCHEMBL30007672 0.76 PAK1 (0.53) AXLCAMKK2PIK3CACYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022237922-A1 ANTITUMOR COMPOUNDS BASED ON NITROGEN HETEROCYCLES AND USE THEREOF AS MEDICAMENTS FAKULTNI NEMOCNICE HRADEC KRALOVE (CZ) 2022-11-17 WO disclosed