SCHEMBL30007692

SCHEMBL30007692

CS(=O)(=O)c1ccc(-c2cnc3[nH]nc(C(=O)O)c3c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 1/20 0.51
GSK3B P49841 1/20 0.51
CAMKK2 Q96RR4 2/20 0.47
PLK4 O00444 2/20 0.45
MAP4K4 O95819 4/20 0.44
MAP4K1 Q92918 1/20 0.43
MINK1 Q8N4C8 3/20 0.43
TNIK Q9UKE5 2/20 0.43
PRKAG1 P54619 1/20 0.43
PRKAA1 Q13131 1/20 0.43
PRKAB1 Q9Y478 1/20 0.43
FYN P06241 1/20 0.43
KCNH2 Q12809 2/20 0.42
PIK3CA P42336 1/20 0.42
PI4KB Q9UBF8 1/20 0.42
MAP2K4 P45985 1/20 0.42
PTGS2 P35354 1/20 0.41
MAPK1 P28482 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30007902 0.87 GSK3A (0.46) GSK3AGSK3BCAMKK2PRKAG1PRKAA1
SCHEMBL30007560 0.78 CA12 (0.43) GSK3AGSK3BMAP4K1PRKAG1PRKAA1
Hydrochloric Acid SCHEMBL30007736 0.78 CAMKK2 (0.57) CAMKK2PIK3CACYP2C9CYP2C19DYRK1B
SCHEMBL4543514 0.76 MAP4K4 (0.52) MAP4K4MINK1TNIKFYNKCNH2
SCHEMBL21225904 0.73 MAP2K4 (0.76) MAP2K4CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL30008041 0.72 CDK5 (0.44) CAMKK2MAP4K4MAP4K1MINK1TNIK
SCHEMBL29623025 0.72 HCAR2 (0.40) PRKAG1PRKAA1PRKAB1MAP2K4MAPK1
SCHEMBL21277005 0.72 HCAR2 (0.40) PRKAG1PRKAA1PRKAB1MAP2K4MAPK1
SCHEMBL30007360 0.71 AXL (0.72) CAMKK2PIK3CACYP2C9CYP2C19DYRK1B
SCHEMBL31072245 0.70 MAP2K4 (0.47) GSK3AGSK3BCAMKK2MAP2K4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022237922-A1 ANTITUMOR COMPOUNDS BASED ON NITROGEN HETEROCYCLES AND USE THEREOF AS MEDICAMENTS FAKULTNI NEMOCNICE HRADEC KRALOVE (CZ) 2022-11-17 WO disclosed