SCHEMBL30007933

SCHEMBL30007933

COc1cc(C(=O)NCC(O)(c2cc(C(C)(C)O)c(F)c(-c3ccc(F)c(F)c3)n2)C2CC2)cc2cc(C)cnc12

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 4/20 0.37
CTSA P10619 5/20 0.36
CNR1 P21554 1/20 0.33
ROCK2 O75116 4/20 0.33
ROCK1 Q13464 4/20 0.33
CYP2C9 P11712 2/20 0.32
MAPK14 Q16539 2/20 0.32
PDE4B Q07343 2/20 0.32
GSK3B P49841 1/20 0.32
BUB1 O43683 1/20 0.31
PRKACG P22612 1/20 0.31
MAPKAPK2 P49137 1/20 0.31
MAPK11 Q15759 1/20 0.31
ACSL5 Q9ULC5 1/20 0.31
STK24 Q9Y6E0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25242930 1.00 GABRA5 (0.37) GABRA5CTSACNR1ROCK2ROCK1
SCHEMBL25687233 1.00 GABRA5 (0.37) GABRA5CTSACNR1ROCK2ROCK1
SCHEMBL30007230 0.93 GABRA5 (0.36) GABRA5CTSACNR1CYP2C9MAPK14
SCHEMBL23958645 0.93 GABRA5 (0.36) GABRA5CTSACNR1CYP2C9MAPK14
SCHEMBL25686195 0.93 GABRA5 (0.36) GABRA5CTSACNR1CYP2C9MAPK14
SCHEMBL30006737 0.93 CNR1 (0.39) GABRA5CTSACNR1ROCK2ROCK1
SCHEMBL25233253 0.93 CNR1 (0.39) GABRA5CTSACNR1ROCK2ROCK1
SCHEMBL25687231 0.93 CNR1 (0.39) GABRA5CTSACNR1ROCK2ROCK1
SCHEMBL25687225 0.93 CFTR (0.35) GABRA5CTSACNR1ROCK2ROCK1
SCHEMBL23958737 0.91 POLB (0.35) ROCK2ROCK1PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461336-A RSV inhibiting 3-substituted quinoline and cinnoline derivatives 爱尔兰詹森科学公司 2022-12-09 CN disclosed