SCHEMBL30006737

SCHEMBL30006737

COc1cc(C(=O)NCC(O)(c2cc(C(C)(C)O)c(F)c(-c3ccc(Cl)cc3)n2)C2CC2)cc2cc(C)cnc12

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.39
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.34
GABRA5 P31644 4/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
CTSA P10619 1/20 0.33
ROCK2 O75116 3/20 0.32
ROCK1 Q13464 3/20 0.32
TP53 P04637 1/20 0.32
RHOC P08134 1/20 0.32
RHOA P61586 1/20 0.32
EGLN1 Q9GZT9 1/20 0.32
S1PR3 Q99500 1/20 0.32
SMPD1 P17405 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25233253 1.00 CNR1 (0.39) CNR1MAPTTHRBGABRA5KDM4E
SCHEMBL25687231 1.00 CNR1 (0.39) CNR1MAPTTHRBGABRA5KDM4E
SCHEMBL25687225 0.94 CFTR (0.35) CNR1MAPTGABRA5ALDH1A1NPSR1
SCHEMBL25687233 0.93 GABRA5 (0.37) CNR1GABRA5CTSAROCK2ROCK1
SCHEMBL30007933 0.93 GABRA5 (0.37) CNR1GABRA5CTSAROCK2ROCK1
SCHEMBL25242930 0.93 GABRA5 (0.37) CNR1GABRA5CTSAROCK2ROCK1
SCHEMBL25687227 0.92 POLB (0.35) MAPTROCK2ROCK1
SCHEMBL23958737 0.92 POLB (0.35) MAPTROCK2ROCK1
SCHEMBL25279914 0.91 CNR1 (0.34) CNR1MAPTGABRA5KDM4EALDH1A1
SCHEMBL30007416 0.91 CNR1 (0.34) CNR1MAPTGABRA5KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461336-A RSV inhibiting 3-substituted quinoline and cinnoline derivatives 爱尔兰詹森科学公司 2022-12-09 CN disclosed