Butorphanol

Butorphanol

SCHEMBL30008734

O=C(O)[C@H](O)[C@@H](O)C(=O)O.Oc1ccc2c(c1)[C@@]13CCCC[C@@]1(O)[C@@H](C2)N(CC1CCC1)CC3

nearest known ligand 0.83

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRK1OPRM1

The experimentally established mechanism targets of Butorphanol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
OPRK1 known ✓ P41145 19/20 0.83
OPRM1 known ✓ P35372 15/20 0.83
OPRD1 P41143 16/20 0.83
KCNH2 Q12809 1/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Butorphanol SCHEMBL41926 1.00 OPRK1 (0.83) OPRK1OPRD1OPRM1KCNH2
Butorphanol SCHEMBL3354253 1.00 OPRK1 (0.83) OPRK1OPRD1OPRM1KCNH2
Butorphanol SCHEMBL30136229 1.00 OPRK1 (0.83) OPRK1OPRD1OPRM1KCNH2
Butorphanol SCHEMBL2727817 1.00 OPRK1 (0.83) OPRK1OPRD1OPRM1KCNH2
Butorphanol SCHEMBL29359664 0.91 OPRK1 (1.00) OPRK1OPRD1OPRM1KCNH2
Butorphanol SCHEMBL20904174 0.91 OPRK1 (1.00) OPRK1OPRD1OPRM1KCNH2
Butorphanol SCHEMBL27701479 0.91 OPRK1 (1.00) OPRK1OPRD1OPRM1KCNH2
Butorphanol SCHEMBL10031253 0.91 OPRK1 (1.00) OPRK1OPRD1OPRM1KCNH2
Butorphanol SCHEMBL16311889 0.91 OPRK1 (1.00) OPRK1OPRD1OPRM1KCNH2
Butorphanol SCHEMBL28094979 0.91 OPRK1 (1.00) OPRK1OPRD1OPRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110545816-B Adhesive patch 久光制药株式会社 2023-04-11 CN disclosed
CN-110573160-B Adhesive patch 久光制药株式会社 2022-11-18 CN disclosed