SCHEMBL30014

SCHEMBL30014

O=C(c1nc2ccc(O)cc2s1)c1cc(O)ccc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 9/20 1.00
HSD17B2 P37059 9/20 1.00
CYP1A2 P05177 2/20 0.65
CYP3A4 P08684 2/20 0.65
CYP2D6 P10635 2/20 0.65
CYP2C9 P11712 2/20 0.65
CYP2B6 P20813 2/20 0.65
CYP2C19 P33261 2/20 0.65
CA12 O43570 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
CA4 P22748 1/20 0.54
CA6 P23280 1/20 0.54
CA5A P35218 1/20 0.54
CA9 Q16790 1/20 0.54
CA14 Q9ULX7 1/20 0.54
CA5B Q9Y2D0 1/20 0.54
MAOB P27338 9/20 0.51
GAA P10253 1/20 0.49
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8403986 0.88 HSD17B1 (0.79) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL8403940 0.88 HSD17B1 (0.78) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL30049 0.84 HSD17B1 (0.76) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL8405368 0.82 HSD17B1 (0.69) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL30246 0.82 HSD17B1 (0.69) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL8400538 0.82 HSD17B1 (0.81) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL29786 0.81 HSD17B1 (1.00) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL4352378 0.80 HSD17B1 (0.67) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL8400525 0.80 HSD17B1 (0.67) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL8401035 0.80 HSD17B1 (0.67) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP claimed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO claimed
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed