SCHEMBL30246

SCHEMBL30246

COc1ccc(O)c(C(=O)c2nc3ccc(OC)cc3s2)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 4/20 0.69
HSD17B2 P37059 4/20 0.69
NPC1 O15118 4/20 0.56
RAB9A P51151 4/20 0.56
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
MAPT P10636 4/20 0.55
MAOB P27338 2/20 0.53
MAOA P21397 1/20 0.53
PDK1 Q15118 1/20 0.52
CYP1A2 P05177 3/20 0.52
CYP3A4 P08684 3/20 0.52
CYP2C19 P33261 3/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
HTT P42858 1/20 0.52
DYRK1A Q13627 1/20 0.52
TSHR P16473 1/20 0.50
HSD17B10 Q99714 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8402838 0.86 HSD17B1 (0.64) HSD17B1HSD17B2NPC1RAB9AMEN1
SCHEMBL30921 0.85 HSD17B1 (0.73) HSD17B1HSD17B2NPC1RAB9AMEN1
SCHEMBL31410 0.85 HSD17B1 (0.73) HSD17B1HSD17B2NPC1RAB9AMEN1
SCHEMBL8404873 0.84 HSD17B1 (0.72) HSD17B1HSD17B2NPC1RAB9AMEN1
SCHEMBL3634489 0.83 HSD17B1 (0.63) HSD17B1HSD17B2NPC1RAB9AMEN1
SCHEMBL30014 0.82 HSD17B1 (1.00) HSD17B1HSD17B2MAPTMAOBCYP1A2
SCHEMBL30687 0.82 HSD17B1 (1.00) HSD17B1HSD17B2NPC1RAB9AMEN1
SCHEMBL8402858 0.82 HSD17B1 (0.69) HSD17B1HSD17B2NPC1RAB9AMEN1
SCHEMBL8405370 0.81 HSD17B1 (0.74) HSD17B1HSD17B2NPC1RAB9AMEN1
SCHEMBL8403873 0.81 HSD17B1 (0.67) HSD17B1HSD17B2NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed