SCHEMBL30015664

SCHEMBL30015664

COc1c(Cl)cc(Br)cc1I

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.35
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
TPMT P51580 3/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34
TUBB4B P68371 1/20 0.34
TUBB3 Q13509 1/20 0.34
TUBB2A Q13885 1/20 0.34
TUBB8 Q3ZCM7 1/20 0.34
TUBA3E Q6PEY2 1/20 0.34
TUBA1A Q71U36 1/20 0.34
TUBA1C Q9BQE3 1/20 0.34
TUBB6 Q9BUF5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19607137 0.84 HSD17B10 (0.45) HSD17B10CA2CA4TPMTKDM4E
SCHEMBL442742 0.84 ALDH1A1 (0.44) HSD17B10CA2CA4TPMTALDH1A1
SCHEMBL23409566 0.78 KMT2A (0.45) HSD17B10CA2TPMTALDH1A1KDM4E
SCHEMBL29970457 0.78 KMT2A (0.45) HSD17B10CA2TPMTALDH1A1KDM4E
SCHEMBL3521150 0.78 HSD17B10 (0.50) HSD17B10CA2CA4TPMTALDH1A1
SCHEMBL30017049 0.77 KDM4E (0.43) HSD17B10CA2CA4TPMTALDH1A1
SCHEMBL19607300 0.77 KDM4E (0.43) HSD17B10CA2CA4TPMTALDH1A1
SCHEMBL931631 0.77 POLB (0.44) HSD17B10CA2CA4TPMTALDH1A1
SCHEMBL20523636 0.75 GAA (0.41) HSD17B10CA2CA4TPMTALDH1A1
SCHEMBL21823580 0.75 TPMT (0.55) HSD17B10CA2CA4TPMTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed