SCHEMBL30016331

SCHEMBL30016331

COc1ccc(Br)cc1S(=N)(=O)c1ccc(C#N)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.46
TSHR P16473 2/20 0.46
GLA P06280 1/20 0.46
GAA P10253 3/20 0.45
ACLY P53396 1/20 0.44
TRPV4 Q9HBA0 1/20 0.43
IDO1 P14902 1/20 0.41
ALOX15 P16050 1/20 0.41
HTT P42858 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ALPL P05186 3/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
EDNRB P24530 2/20 0.39
EDNRA P25101 2/20 0.39
WDR5 P61964 1/20 0.39
KDM4E B2RXH2 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21760971 0.78 SMN1; SMN2 (0.48) SMN1; SMN2TSHRGLAGAATRPV4
SCHEMBL29134947 0.78 ALPL (0.58) SMN1; SMN2GLAALPLKMT2A
SCHEMBL30909386 0.73 TRPV4 (0.45) ACLYTRPV4IDO1ALPL
SCHEMBL30015429 0.72 IDO1 (0.43) IDO1CA12CA1CA2CA9
SCHEMBL1790129 0.70 SMN1; SMN2 (0.65) SMN1; SMN2TSHRGLAGAAALOX15
SCHEMBL30514814 0.70 SMN1; SMN2 (0.65) SMN1; SMN2TSHRGLAGAAALOX15
SCHEMBL13211338 0.69 SMN1; SMN2 (0.59) SMN1; SMN2ACLYTRPV4ALPL
SCHEMBL47015 0.69 SMN1; SMN2 (0.64) SMN1; SMN2TSHRGLAGAATRPV4
SCHEMBL1137871 0.69 SMN1; SMN2 (0.59) SMN1; SMN2TSHRGLAGAAALOX15
SCHEMBL7421633 0.69 SMN1; SMN2 (0.59) SMN1; SMN2TSHRGLAGAAACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed