SCHEMBL30016751

SCHEMBL30016751

CC1(C)OB(c2ccc3c(=O)[nH]cnc3c2)OC1(C)C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.54
CHEK1 O14757 2/20 0.54
PIM1 P11309 2/20 0.54
RPS6KA3 P51812 1/20 0.54
ALDH1A1 P00352 1/20 0.50
PIK3CD O00329 1/20 0.44
PIK3CA P42336 1/20 0.44
PIK3CB P42338 1/20 0.44
PDPK1 O15530 1/20 0.44
CA12 O43570 1/20 0.44
ALOX15 P16050 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CA9 Q16790 1/20 0.44
TNKS2 Q9H2K2 1/20 0.44
PRMT5 O14744 2/20 0.42
WDR77 Q9BQA1 2/20 0.42
KDM4A O75164 1/20 0.41
KDM4B O94953 1/20 0.41
KDM5C P41229 1/20 0.41
KDM4C Q9H3R0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL393560 1.00 PARP1 (0.54) PARP1CHEK1PIM1RPS6KA3ALDH1A1
SCHEMBL8212169 0.89 PARP1 (0.54) PARP1CHEK1PIM1RPS6KA3PDPK1
SCHEMBL2379179 0.80 LPL (0.40) ALDH1A1CA9LPLLIPG
SCHEMBL3263058 0.78 PRMT5 (0.40) CA12CA9PRMT5WDR77LPL
SCHEMBL31037319 0.77 KDM4E (0.48) PARP1ALDH1A1SMN1; SMN2TNKS2PRMT5
SCHEMBL3263196 0.77 KDM4E (0.48) PARP1ALDH1A1SMN1; SMN2TNKS2PRMT5
SCHEMBL29525463 0.77 MMP12 (0.45) LPLLIPG
SCHEMBL874992 0.77 MMP12 (0.45) LPLLIPG
SCHEMBL391998 0.75 GSK3A (0.46) PARP1CHEK1PIM1RPS6KA3ALDH1A1
SCHEMBL3225882 0.75 PRMT5 (0.40) CA12CA9PRMT5WDR77LPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed