SCHEMBL24698161

SCHEMBL24698161

N#Cc1ccc(-c2nc(N3CCC3)nc3c2CCC3)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 3/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
KDM4E B2RXH2 3/20 0.36
ADORA2A P29274 2/20 0.36
EGLN2 Q96KS0 1/20 0.35
IGF1R P08069 2/20 0.35
ALDH1A1 P00352 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
AR P10275 1/20 0.34
NSD2 O96028 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24699042 0.86 CYP11B2 (0.48) CYP11B2KDM4EADORA2A
SCHEMBL24698160 0.84 AR (0.36) CYP11B2KDM4EEGLN2ALDH1A1HPGD
SCHEMBL30016865 0.84 AR (0.36) CYP11B2KDM4EEGLN2ALDH1A1HPGD
SCHEMBL24699497 0.83 HSD17B10 (0.43) KDM4EALDH1A1SMN1; SMN2MAPTHPGD
SCHEMBL24699459 0.79 GBA1 (0.39) KDM4EIGF1RALDH1A1MAPTHPGD
SCHEMBL24699158 0.78 IGF1R (0.34) KDM4EIGF1RALDH1A1SMN1; SMN2MAPT
SCHEMBL24697795 0.75 ALDH1A1 (0.40) KDM4EIGF1RALDH1A1SMN1; SMN2MAPT
SCHEMBL24699477 0.75 ALDH1A1 (0.47) KDM4EIGF1RALDH1A1MAPTHPGD
SCHEMBL24698171 0.74 ALDH1A1 (0.54) KDM4EALDH1A1SMN1; SMN2MAPTHPGD
SCHEMBL24697814 0.74 HRH3 (0.44) ALDH1A1SMN1; SMN2HTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed