SCHEMBL30030003

SCHEMBL30030003

NC(=O)c1cccc(-c2ccc(N)cc2)c1I

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.50
PARP1 P09874 3/20 0.46
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
IKBKB O14920 2/20 0.38
GRK6 P43250 1/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PDCD1 Q15116 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
HNF4A P41235 1/20 0.36
CHEK1 O14757 1/20 0.35
ALOX5AP P20292 1/20 0.35
FEN1 P39748 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8102370 0.86 BCAT2 (0.69) BCAT2PARP1KEAP1NFE2L2IKBKB
SCHEMBL28053360 0.85 BCAT2 (0.49) BCAT2KEAP1NFE2L2IKBKBKDM4E
SCHEMBL3791160 0.82 BCAT2 (0.53) BCAT2PARP1KEAP1NFE2L2MKNK1
SCHEMBL1982663 0.82 BCAT2 (0.74) BCAT2PARP1KEAP1NFE2L2MKNK1
SCHEMBL27895562 0.81 BCAT2 (0.52) BCAT2PARP1KEAP1NFE2L2MKNK1
SCHEMBL17143067 0.79 BCAT2 (0.50) BCAT2PARP1KEAP1NFE2L2MKNK1
SCHEMBL27895561 0.78 BCAT2 (0.53) BCAT2PARP1KEAP1NFE2L2MKNK1
SCHEMBL30029239 0.78 EIF4E (0.46) BCAT2PARP1KEAP1NFE2L2MKNK1
SCHEMBL27486058 0.77 KDM4E (0.52) BCAT2PARP1KEAP1NFE2L2KDM4E
SCHEMBL31682597 0.76 BCAT2 (0.44) BCAT2PARP1IKBKBGRK6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113831302-B Benzisoselenazolone derivative and preparation method and application thereof 山东大学 2022-11-29 CN disclosed