SCHEMBL300340

SCHEMBL300340

CC1(OC(=O)N2CC[C@H](Oc3cc(Cl)ncn3)C(F)C2)CC1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 15/20 0.40
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
TBK1 Q9UHD2 5/20 0.35
JAK2 O60674 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL759976 1.00 GPR119 (0.40) GPR119CYP2C9CYP2C19TBK1JAK2
SCHEMBL298847 1.00 GPR119 (0.40) GPR119CYP2C9CYP2C19TBK1JAK2
SCHEMBL288238 0.83 GPR119 (0.55) GPR119CYP2C9CYP2C19
SCHEMBL10170824 0.82 GPR119 (0.42) GPR119CYP2C9CYP2C19
SCHEMBL1768452 0.82 GPR119 (0.42) GPR119CYP2C9CYP2C19
SCHEMBL1768451 0.82 GPR119 (0.42) GPR119CYP2C9CYP2C19
SCHEMBL756571 0.77 GPR119 (0.39) GPR119CYP2C9CYP2C19TBK1JAK2
SCHEMBL299860 0.77 GPR119 (0.39) GPR119CYP2C9CYP2C19TBK1JAK2
SCHEMBL298683 0.77 GPR119 (0.38) GPR119CYP2C9CYP2C19TBK1JAK2
SCHEMBL756824 0.77 GPR119 (0.38) GPR119CYP2C9CYP2C19TBK1JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427450-A1 GPR 119 MODULATORS Pfizer Inc. (US) 2012-03-14 EP disclosed
EP-2427448-A1 Gpr 119 modulators Pfizer Inc. (US) 2012-03-14 EP disclosed