SCHEMBL300505

SCHEMBL300505

C[C@H](NC(=O)c1nn(Cc2ccccc2)c2c1CCCCC2)C1CCCCC1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.46
CNR2 P34972 3/20 0.46
CNR1 P21554 2/20 0.46
EPHX2 P34913 2/20 0.45
RIPK1 Q13546 1/20 0.45
ALDH1A1 P00352 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
PPARG P37231 1/20 0.41
BRD4 O60885 1/20 0.41
TACR2 P21452 3/20 0.41
TACR3 P29371 3/20 0.41
OPRM1 P35372 2/20 0.41
SMYD3 Q9H7B4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14003141 1.00 SIGMAR1 (0.46) SIGMAR1CNR2CNR1EPHX2RIPK1
SCHEMBL14003143 1.00 SIGMAR1 (0.46) SIGMAR1CNR2CNR1EPHX2RIPK1
SCHEMBL2715441 0.88 MEN1 (0.41) SIGMAR1CNR2CNR1RIPK1ALDH1A1
SCHEMBL13871389 0.84 ALDH1A1 (0.58) SIGMAR1CNR2CNR1EPHX2ALDH1A1
SCHEMBL13871545 0.84 CNR1 (0.43) CNR2CNR1EPHX2RIPK1ALDH1A1
SCHEMBL300548 0.83 EPHX2 (0.43) SIGMAR1EPHX2ALDH1A1SMN1; SMN2BRD4
SCHEMBL300503 0.83 EPHX2 (0.43) SIGMAR1EPHX2ALDH1A1SMN1; SMN2BRD4
SCHEMBL13889613 0.83 ALDH1A1 (0.53) CNR2CNR1ALDH1A1MEN1KMT2A
SCHEMBL14003140 0.83 ALDH1A1 (0.53) CNR2CNR1ALDH1A1MEN1KMT2A
SCHEMBL13871582 0.83 SIGMAR1 (0.43) SIGMAR1CNR2CNR1EPHX2RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937259-B1 HEXAHYDRO-CYCLOHEPTAPYRAZOLE CANNABINOID MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-11-23 EP claimed