SCHEMBL30065560

SCHEMBL30065560

COc1cc(NC(=O)c2cc(Cl)c(C(F)(F)F)cc2Cc2ccc(F)cc2C)ccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SORT1 Q99523 2/20 0.48
SCN10A Q9Y5Y9 3/20 0.43
HDAC4 P56524 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
RET P07949 2/20 0.39
KDR P35968 3/20 0.39
BRAF P15056 3/20 0.38
AURKB Q96GD4 2/20 0.38
RAF1 P04049 2/20 0.38
MEN1 O00255 1/20 0.38
PLK4 O00444 1/20 0.38
CIT O14578 1/20 0.38
AURKA O14965 1/20 0.38
MUSK O15146 1/20 0.38
EPHB6 O15197 1/20 0.38
MAPK13 O15264 1/20 0.38
MLNR O43193 1/20 0.38
MAP3K7 O43318 1/20 0.38
RIPK2 O43353 1/20 0.38
DYRK3 O43781 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28651365 1.00 SORT1 (0.48) SORT1SCN10AHDAC4HDAC6RET
SCHEMBL28669416 0.88 SORT1 (0.45) SORT1SCN10AHDAC4HDAC6RET
SCHEMBL30065594 0.88 SORT1 (0.45) SORT1SCN10AHDAC4HDAC6RET
SCHEMBL28928647 0.85 SORT1 (0.62) SORT1SCN10AHDAC4HDAC6
SCHEMBL30065536 0.85 SORT1 (0.62) SORT1SCN10AHDAC4HDAC6
SCHEMBL22942187 0.83 SCN8A (0.49) SORT1SCN10A
SCHEMBL22941942 0.81 SORT1 (0.58) SORT1SCN10AHDAC4HDAC6RET
SCHEMBL22942186 0.80 SCN8A (0.47) SORT1SCN10AKDRRAF1MET
SCHEMBL22203188 0.80 BRAF (0.38) SCN10AKDRBRAF
SCHEMBL29435940 0.80 BRAF (0.38) SCN10AKDRBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112996774-B 2-oxo-1,2-dihydropyridine derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-11-22 CN disclosed