SCHEMBL30099343

SCHEMBL30099343

Brc1ccc2c(Br)cncc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 2/20 0.39
METAP2 P50579 2/20 0.39
CSNK2A1 P68400 1/20 0.39
CYP2A6 P11509 2/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
BACE1 P56817 2/20 0.35
DYRK1A Q13627 1/20 0.35
PLAU P00749 1/20 0.35
PDPK1 O15530 1/20 0.34
JAK2 O60674 1/20 0.34
CHUK O15111 1/20 0.34
ERN1 O75460 1/20 0.34
ACHE P22303 1/20 0.34
NPM1 P06748 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5497704 1.00 NOS1 (0.39) NOS1METAP2CSNK2A1CYP2A6CYP11B1
SCHEMBL20423421 0.79 HSD17B1 (0.42) CYP11B1CYP11B2KDM4EMEN1ALDH1A1
SCHEMBL20975068 0.79 CYP11B2 (0.37) CYP2A6CYP11B1CYP11B2MAPTBACE1
SCHEMBL30804194 0.79 NOS1 (0.37) NOS1METAP2CSNK2A1CYP2A6CYP11B1
SCHEMBL29709757 0.79 NOS1 (0.37) NOS1CYP2A6DYRK1ACHUKACHE
SCHEMBL4306327 0.79 CYP1A2 (0.41) CYP2A6KDM4EALDH1A1BACE1ACHE
SCHEMBL4064559 0.79 NOS1 (0.37) NOS1CYP2A6DYRK1ACHUKACHE
SCHEMBL13172306 0.79 ERN1 (0.43) NOS1METAP2CSNK2A1CYP2A6CYP11B1
SCHEMBL28716125 0.79 NOS1 (0.37) NOS1METAP2CSNK2A1CYP2A6CYP11B1
SCHEMBL30572689 0.79 NPM1 (0.39) NOS1METAP2CSNK2A1CYP2A6CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110612294-B Human cerebulin ligands and bifunctional compounds comprising same 阿尔维纳斯运营股份有限公司 2024-01-16 CN disclosed
CN-115974840-A Human cereblon ligand and bifunctional compound comprising same 阿尔维纳斯运营股份有限公司 2023-04-18 CN disclosed
WO-2022251359-A1 BICYCLIC INHIBITORS OF ALK5 AND METHODS OF USE THERAVANCE BIOPHARMA R&D IP, LLC (US) 2022-12-01 WO disclosed