SCHEMBL30107343

SCHEMBL30107343

COc1ccc(Cn2cncc2C2(C(=O)O)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 9/20 0.53
CYP11B1 P15538 8/20 0.53
HSP90AA1 P07900 1/20 0.44
HSP90AB1 P08238 1/20 0.44
CACNA1G O43497 1/20 0.43
CACNA1H O95180 1/20 0.43
CACNA1I Q9P0X4 1/20 0.43
CYP19A1 P11511 1/20 0.42
ALDH1A1 P00352 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
IDO1 P14902 1/20 0.40
GABRA5 P31644 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23535858 0.72 CYP11B2 (0.58) CYP11B2CYP11B1HSP90AA1HSP90AB1CYP19A1
SCHEMBL20519574 0.72 CYP11B1 (0.54) CYP11B2CYP11B1HSP90AA1HSP90AB1CYP19A1
SCHEMBL20524347 0.72 CYP11B1 (0.54) CYP11B2CYP11B1HSP90AA1HSP90AB1CYP19A1
SCHEMBL20519343 0.71 CYP11B1 (0.51) CYP11B2CYP11B1HSP90AA1HSP90AB1CYP19A1
SCHEMBL30107166 0.71 CYP11B1 (0.51) CYP11B2CYP11B1HSP90AA1HSP90AB1CYP19A1
SCHEMBL6929673 0.71 CYP11B1 (0.75) CYP11B2CYP11B1HSP90AA1HSP90AB1IDO1
SCHEMBL15507125 0.70 CYP11B1 (0.61) CYP11B2CYP11B1HSP90AA1HSP90AB1CYP19A1
SCHEMBL31138699 0.70 CYP11B1 (0.56) CYP11B2CYP11B1HSP90AA1HSP90AB1CYP19A1
SCHEMBL28941444 0.70 CYP11B1 (0.61) CYP11B2CYP11B1HSP90AA1HSP90AB1CYP19A1
SCHEMBL8129319 0.70 CYP11B2 (0.62) CYP11B2CYP11B1HSP90AA1HSP90AB1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110678466-B Diazanaphthalenes as HPK1 inhibitors 豪夫迈·罗氏有限公司 2023-01-31 CN disclosed