SCHEMBL30120157

SCHEMBL30120157

CC(C)(C)OC(=O)N1CCN(CCn2cnc3ccc(Oc4c(F)ccc(F)c4C#N)cc3c2=O)CC1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRAF P15056 3/20 0.47
ENPP2 Q13822 7/20 0.42
SQOR Q9Y6N5 1/20 0.40
IDO1 P14902 1/20 0.40
TDO2 P48775 1/20 0.40
IDO2 Q6ZQW0 1/20 0.40
PLK1 P53350 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.38
NSD2 O96028 1/20 0.37
GPR119 Q8TDV5 1/20 0.37
BTK Q06187 1/20 0.37
P2RX3 P56373 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24542773 1.00 BRAF (0.47) BRAFENPP2SQORIDO1TDO2
SCHEMBL24542899 0.91 BRAF (0.46) BRAFENPP2SQORIDO1TDO2
SCHEMBL30120168 0.89 BRAF (0.46) BRAFENPP2IRAK4GPR119BTK
SCHEMBL26591137 0.89 BRAF (0.46) BRAFENPP2IRAK4GPR119BTK
SCHEMBL29743471 0.89 BRAF (0.54) BRAFENPP2SQORIDO1TDO2
SCHEMBL24542883 0.89 BRAF (0.54) BRAFENPP2SQORIDO1TDO2
SCHEMBL29743396 0.89 BRAF (0.52) BRAFENPP2SQORIDO1TDO2
SCHEMBL26185967 0.89 BRAF (0.52) BRAFENPP2SQORIDO1TDO2
SCHEMBL30120453 0.89 GPR119 (0.46) BRAFENPP2IRAK4GPR119BTK
SCHEMBL29196989 0.89 GPR119 (0.46) BRAFENPP2IRAK4GPR119BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4263518-B1 NEW QUINAZOLINONE DERIVATIVES HOFFMANN LA ROCHE (CH) 2026-04-01 EP disclosed
US-12570615-B2 Quinazolinone derivatives HOFFMANN-LA ROCHE INC. 2026-03-10 US disclosed
EP-4351583-A1 THERAPEUTICS FOR THE DEGRADATION OF MUTANT BRAF C4 Therapeutics, Inc. (US) 2024-04-17 EP disclosed
US-20230331682-A1 NEW QUINAZOLINONE DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 2023-10-19 US disclosed
WO-2022261250-A1 THERAPEUTICS FOR THE DEGRADATION OF MUTANT BRAF C4 THERAPEUTICS, INC. (US) 2022-12-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230331682-A1 NEW QUINAZOLINONE DERIVATIVES NDUFS3, NQO2, NDUFC1 BRAF 2269/4885ENPP2 3402/4885SQOR 88/4885
US-12570615-B2 Quinazolinone derivatives ABL1, NQO2, CNR1 BRAF 1372/4885ENPP2 2484/4885SQOR 974/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.