SCHEMBL30120770

SCHEMBL30120770

COc1ccc(Cl)c(Cl)c1C1CCC(COS(=O)(=O)c2ccc(C)cc2)N1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
HTR2B P41595 2/20 0.38
ALDH1A1 P00352 7/20 0.37
GAA P10253 5/20 0.37
TSHR P16473 4/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
POLB P06746 1/20 0.37
KDM4E B2RXH2 2/20 0.35
GLA P06280 1/20 0.35
HPGD P15428 1/20 0.35
RUNX1 Q01196 1/20 0.35
ATM Q13315 1/20 0.35
CBFB Q13951 1/20 0.35
RCE1 Q9Y256 1/20 0.35
APEX1 P27695 1/20 0.35
PKM P14618 1/20 0.35
MAPT P10636 1/20 0.35
THRB P10828 1/20 0.35
DRD2 P14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30121107 0.89 HTR2A (0.38) HTR2AHTR2CHTR2BALDH1A1GAA
SCHEMBL30120779 0.81 HTR2A (0.45) HTR2AHTR2CHTR2BDRD2
SCHEMBL23217487 0.81 HTR2A (0.38) HTR2AHTR2CHTR2BALDH1A1GAA
SCHEMBL30120952 0.79 HTR2A (0.45) HTR2AHTR2CHTR2BGLADRD2
SCHEMBL18396809 0.79 STAT3 (0.45) ALDH1A1POLBKDM4EKMT2ACYP1A2
SCHEMBL30120868 0.78 HTR2A (0.42) HTR2AHTR2CHTR2BDRD2
SCHEMBL30120802 0.76 FFAR2 (0.47) HTR2AHTR2CHTR2B
SCHEMBL2463859 0.74 STAT3 (0.41) ALDH1A1TSHRPOLBMAPTKMT2A
SCHEMBL29844877 0.73 HTR2A (0.37) HTR2AHTR2CHTR2BALDH1A1GAA
SCHEMBL2462885 0.71 CYP2C19 (0.43) ALDH1A1TSHRPOLBKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313313-A1 ARYL HETEROCYCLIC COMPOUNDS AS KV1.3 POTASSIUM SHAKER CHANNEL BLOCKERS D.E. Shaw Research, LLC (US) 2024-02-07 EP disclosed
WO-2022212296-A1 ARYL HETEROCYCLIC COMPOUNDS AS Kv1.3 POTASSIUM SHAKER CHANNEL BLOCKERS D.E. SHAW RESEARCH, LLC (US) 2022-10-06 WO disclosed