SCHEMBL30120802

SCHEMBL30120802

COc1ccc(Cl)c(Cl)c1C1CCC(C(=O)O)N1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FFAR2 O15552 18/20 0.47
HTR2A P28223 2/20 0.45
HTR2C P28335 2/20 0.45
HTR2B P41595 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30120779 0.84 HTR2A (0.45) FFAR2HTR2AHTR2CHTR2B
SCHEMBL30120952 0.81 HTR2A (0.45) FFAR2HTR2AHTR2CHTR2B
SCHEMBL30120868 0.80 HTR2A (0.42) FFAR2HTR2AHTR2CHTR2B
SCHEMBL23217560 0.79 HTR2A (0.42) FFAR2HTR2AHTR2CHTR2B
SCHEMBL23217172 0.79 HTR2C (0.44) FFAR2HTR2AHTR2CHTR2B
SCHEMBL23217480 0.79 HTR2C (0.44) FFAR2HTR2AHTR2CHTR2B
SCHEMBL30120770 0.76 HTR2A (0.38) HTR2AHTR2CHTR2B
SCHEMBL30721088 0.74 ALDH1A1 (0.43) HTR2AHTR2CHTR2B
SCHEMBL30721081 0.74 ALDH1A1 (0.43) HTR2AHTR2CHTR2B
SCHEMBL23214520 0.73 HTR2A (0.41) FFAR2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313313-A1 ARYL HETEROCYCLIC COMPOUNDS AS KV1.3 POTASSIUM SHAKER CHANNEL BLOCKERS D.E. Shaw Research, LLC (US) 2024-02-07 EP disclosed
WO-2022212296-A1 ARYL HETEROCYCLIC COMPOUNDS AS Kv1.3 POTASSIUM SHAKER CHANNEL BLOCKERS D.E. SHAW RESEARCH, LLC (US) 2022-10-06 WO disclosed