SCHEMBL30131343

SCHEMBL30131343

O=C(NCC1CC(F)(F)C1)c1ncccc1Cl

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 9/20 0.51
IL1B P01584 7/20 0.44
CNR1 P21554 6/20 0.42
CNR2 P34972 6/20 0.42
KDM1A O60341 1/20 0.41
KCNA5 P22460 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30131489 0.83 P2RX7 (0.58) P2RX7CNR1CNR2
SCHEMBL30250478 0.80 MAPT (0.54) P2RX7
SCHEMBL30875023 0.79 P2RX7 (0.48) P2RX7CNR1CNR2KCNA5PDE4A
SCHEMBL31275734 0.77 P2RX7 (0.41) P2RX7
SCHEMBL20068866 0.77 SSTR4 (0.49) P2RX7CNR1CNR2
SCHEMBL20147919 0.76 HTR4 (0.45) P2RX7CNR1CNR2
SCHEMBL30875055 0.74 EGLN2 (0.44)
SCHEMBL20158754 0.73 RET (0.45) P2RX7CNR1CNR2
SCHEMBL30131408 0.73 NPC1 (0.47) PDE4APDE4BPDE4CPDE4D
SCHEMBL30875025 0.72 ALDH1A1 (0.43) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117715898-A Six-membered aryl or heteroaryl amide compound, composition and application thereof 贝达药业股份有限公司 2024-03-15 CN claimed
WO-2023279986-A1 SIX-MEMBERED ARYL OR HETEROARYL AMIDES, AND COMPOSITION AND USE THEREOF 贝达药业股份有限公司 2023-01-12 WO claimed
CN-117715898-A Six-membered aryl or heteroaryl amide compound, composition and application thereof 贝达药业股份有限公司 2024-03-15 CN disclosed
WO-2023279986-A1 SIX-MEMBERED ARYL OR HETEROARYL AMIDES, AND COMPOSITION AND USE THEREOF 贝达药业股份有限公司 2023-01-12 WO disclosed